BDBM725750 US20250074910, Example 47-1

SMILES CC(C)N(C(=O)c1cc(F)ccc1Oc1nncnc1N1CC2(CCN(CC3CCC4(CC3)CC(=O)N(C)C4)CC2)C1)C(C)C

InChI Key InChIKey=MAJPYCXXBJRPIF-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 725750   

TargetHistone-lysine N-methyltransferase 2A(Human)
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US Patent
LigandPNGBDBM725750(US20250074910, Example 47-1)
Affinity DataIC50: 20.2nMAssay Description:The inhibition of Menin/MLL-4-43 peptide interaction by small molecule inhibitors was quantitatively detected by fluorescence polarization competitio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/9/2025
Entry Details
US Patent