BDBM727089 US12252493, Example 39

SMILES Cc1ncccc1-c1cnc(NCc2c(F)ccc3c2CCO3)n2cc(C(C)N)nc12

InChI Key InChIKey=LOBZJLAGRIYYGQ-UHFFFAOYSA-N

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 727089   

TargetHistone-binding protein RBBP4/Histone-lysine N-methyltransferase EZH2/Polycomb protein EED/Polycomb protein SUZ12/Zinc finger protein AEBP2(Human)
Mirati Therapeutics

US Patent

LigandBDBM727089(US12252493, Example 39)Copy SMILESCopy InChI

Affinity DataIC50: 250nMAssay Description:Briefly, compounds of the present invention were solubilized in DMSO and a series of 10, three-fold serial dilutions were made for each compound in 1...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In Depth
Date in BDB:
7/22/2025
Entry Details
Copy BDB DOIUS Patent

Copy reaction URL