BDBM728181 2-benzyl-2-azaspiro [3.3]heptan-6-yl (2R)-4-[5- (cyclopropanesulfonyl) pyrimidin-2-yl]-2- methylpiperazine-1- carboxylate::US20250092022, Compound 22

SMILES C[C@@H]1CN(c2ncc(S(=O)(=O)C3CC3)cn2)CCN1C(=O)OC1CC2(C1)CN(Cc1ccccc1)C2

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 728181   

TargetMuscarinic acetylcholine receptor M4(Human)
Neurocrine Biosciences

US Patent
LigandPNGBDBM728181(2-benzyl-2-azaspiro [3.3]heptan-6-yl (2R)-4-[5- (c...)
Affinity DataKi: <100nMAssay Description:Binding affinity (Ki) for the compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M4 receptor. M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/25/2025
Entry Details
US Patent