BDBM730781 US20250122182, Syn. Ex. 102

SMILES C=C(F)C(=O)NCc1cnn(Cc2cc(OC)c3c(NS(=O)(=O)c4cc(CC)ccc4OCCNC(=O)OCC4c5ccccc5C5C=CC=CC54)noc3c2)c1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 730781   

TargetHistone acetyltransferase KAT6A(Human)
Isosterix

US Patent
LigandPNGBDBM730781(US20250122182, Syn. Ex. 102)
Affinity DataIC50: 2nMAssay Description:The Kat6a inhibitory activity of test compounds was determined using an Alpha Screen-based detection method. The assay reactions were conducted in a ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetHistone acetyltransferase KAT6B(Human)
Isosterix

US Patent
LigandPNGBDBM730781(US20250122182, Syn. Ex. 102)
Affinity DataIC50: 2.53E+3nMAssay Description:The Kat6a inhibitory activity of test compounds was determined using an Alpha Screen-based detection method. The assay reactions were conducted in a ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent