BDBM732081 (R)-3-((1R,3R)-1-(2,6- difluoro-4-((1-(3- fluoropropyl)azetidin-3- yl)amino)phenyl)-5-fluoro-3- methyl-3,4-dihydro-1H- pyrido[3,4-b]indol-2(9H)-yl)- 2-fluoro-2-methylpropan-1-ol::US20250114338, Example 400

SMILES C[C@@H]1Cc2c([nH]c3cccc(F)c23)[C@@H](c2c(F)cc(NC3CN(CCCF)C3)cc2F)N1C[C@@](C)(F)CO

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 732081   

TargetEstrogen receptor(Human)
Genentech

US Patent
LigandPNGBDBM732081((R)-3-((1R,3R)-1-(2,6- difluoro-4-((1-(3- fluoropr...)
Affinity DataEC50:  0.0230nMAssay Description:All of the exemplary Formula I compounds in Tables 1 and 2 were tested for binding to ERa (Estrogen Receptor alpha) and biological activity according...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Date in BDB:
8/22/2025
Entry Details
US Patent