BDBM732842 5-[4-carbamoyl-5-methoxy-2-[(3S)-3- (morpholinomethyl)-3,4-dihydro-1H- isoquinoline-2-carbonyl]phenyl]-N-(4- chlorophenyl)-N-[(2- methoxyphenyl)methyl]-1,2-dimethyl- pyrrole-3-carboxamide::US20250115577, Compound 63

SMILES COc1ccccc1CN(C(=O)c1cc(-c2cc(OC)c(C(N)=O)cc2C(=O)N2Cc3ccccc3C[C@H]2CN2CCOCC2)n(C)c1C)c1ccc(Cl)cc1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 732842   

TargetApoptosis regulator Bcl-2(Human)
Eil Therapeutics

US Patent
LigandPNGBDBM732842(5-[4-carbamoyl-5-methoxy-2-[(3S)-3- (morpholinomet...)
Affinity DataIC50: 30nMAssay Description:BPS Bioscience, #50222: 3 ng of BCL-2, 5 μL of 1:100 anti-His Tb-labeled donor, 5 μL of 1:100 Dye-labeled acceptor, 5 L of 1:40 BCL-2 Peptide Ligand,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
US Patent