BDBM736281 N-methyl-2-(2-((1-methyl-9- (1-methyl-1H-pyrazol-4-yl)-6,7-dihydro- 5H-benzo[c][1,2,3]triazolo[1,5-a] azepin-7-yl)amino)phenyl)acetamide::US12286435, Code LC11

SMILES CNC(=O)Cc1ccccc1NC1CCn2nnc(C)c2-c2ccc(-c3cnn(C)c3)cc21

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 736281   

TargetBromodomain-containing protein 4 [58-164](Human)
Bionna (Beijing) Medical Technology

US Patent
LigandPNGBDBM736281(N-methyl-2-(2-((1-methyl-9- (1-methyl-1H-pyrazol-...)
Affinity DataKi:  7.80nMAssay Description:The purity of BRD4 BD1 protein used in the experiment was greater than 95%, and the protein concentration was 43.4 uM. The 96-well plate was purchase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/28/2025
Entry Details
US Patent