BDBM736805 US20250136577, Example 31

SMILES CN1C2C(Br)=CN=CC2N(C(=O)NC2C=NC(n3nccn3)=C(Cl)C2)CC1(C)C

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 736805   

LigandPNGBDBM736805(US20250136577, Example 31)
Affinity DataIC50: 260nMAssay Description:MALT1 protease activity was assessed in vitro by measuring the cleavage of a fluorogenic tetrapeptide substrate.For a higher sensitivity assay, comme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM736805(US20250136577, Example 31)
Affinity DataIC50: 3.00E+3nMAssay Description:MALT1 protease activity was assessed in vitro by measuring the cleavage of a fluorogenic tetrapeptide substrate.[0581]A protein (MALT1-GS-Ub) compris...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent