BDBM736808 US20250136577, Example 34
SMILES CC[C@@H]1CN(C(=O)Nc2cnc(-n3nccn3)c(Cl)c2)c2cncc(Br)c2N1C
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 736808
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1 [339-715](Human)
C4X Discovery
US Patent
C4X Discovery
US Patent
Affinity DataIC50: 50nMAssay Description:MALT1 protease activity was assessed in vitro by measuring the cleavage of a fluorogenic tetrapeptide substrate.For a higher sensitivity assay, comme...More data for this Ligand-Target Pair
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1 [339-715](Human)
C4X Discovery
US Patent
C4X Discovery
US Patent
Affinity DataIC50: 970nMAssay Description:MALT1 protease activity was assessed in vitro by measuring the cleavage of a fluorogenic tetrapeptide substrate.[0581]A protein (MALT1-GS-Ub) compris...More data for this Ligand-Target Pair
