BDBM736817 US20250136577, Example 43
SMILES Cc1ncc2c(c1Br)O[C@H](C(F)(F)F)CN2C(=O)NC1C=NC(n2nccn2)=C(Cl)C1
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 736817
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1 [339-715](Human)
C4X Discovery
US Patent
C4X Discovery
US Patent
Affinity DataIC50: 60nMAssay Description:MALT1 protease activity was assessed in vitro by measuring the cleavage of a fluorogenic tetrapeptide substrate.For a higher sensitivity assay, comme...More data for this Ligand-Target Pair
