BDBM739049 US20250145633, Example 298
SMILES COc1ccc(C2(NC(=O)c3c(C)oc4ncnc(NC5(C)CC5)c34)CC2)cc1F
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 739049
TargetDual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B(Human)
Dart Neuroscience
US Patent
Dart Neuroscience
US Patent
Affinity DataIC50: 10nMAssay Description:PDE1B inhibition was determined by an IMAP TR-FRET assay. The IMAP TR-FRET PDE assay was optimized for concentration of enzyme, Calmodulin, cAMP or c...More data for this Ligand-Target Pair
