BDBM741323 COT-PEG4- triazole-P8::US20250161476, LP# LP10

SMILES CCc1cc(OCCCCn2cc(COCCOCCOCCOCCNC(=O)COC3C#CCCCCC3)nn2)ccc1-c1ccc(C[C@H](NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@](C)(Cc2ccccc2F)NC(=O)[C@@H](NC(=O)CNC(=O)[C@H](Cc2nn[nH]n2)NC(=O)C(C)(C)C(=O)NCCc2cnc[nH]2)[C@@H](C)O)[C@@H](C)O)C(=O)N[C@@H](CCCc2cc(C)cc(C)c2)C(N)=O)cc1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 741323   

TargetGlucagon-like peptide 1 receptor(Human)
Regeneron Pharmaceuticals

US Patent
LigandPNGBDBM741323(COT-PEG4- triazole-P8 | US20250161476, LP# LP10)
Affinity DataEC50:  0.982nMAssay Description:For the assay, HEK293 cells over-expressing full length human GLP-1R were utilized and the downstream cAMP accumulation was assessed as a measure of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/19/2025
Entry Details
US Patent