BDBM743394 1-[6-[5-[6-[4-[2-(2,6-dioxo-3-piperidyl)-1-oxo-isoindolin-5-yl]piperazin-1-yl]-6-oxo- hexyl]-1,2,4-oxadiazol-3-yl]-5-(trifluoromethyl)-3-pyridyl]-3-(7- isopropylpyrazolo[1,5-a]pyrimidin-6-yl)urea::US20250163066, Compound 162

SMILES CC(C)c1c(NC(=O)Nc2cnc(-c3noc(CCCCCC(=O)N4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)n3)c(C(F)(F)F)c2)cnc2ccnn12

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 743394   

LigandPNGBDBM743394(1-[6-[5-[6-[4-[2-(2,6-dioxo-3-piperidyl)-1-oxo-iso...)
Affinity DataEC50: <200nMAssay Description:Compound activity was determined using recombinant MALT1 protein (Creative Biomart, Cat #MALT1-28H) and Ac-LRSR-AMC Substrate in an in vitro enzymati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/20/2025
Entry Details
US Patent