BDBM748437 US20250188030, Compound C18

SMILES CCc1c(F)cccc1-c1cc(C(C)(C)C(=O)NS(=O)(=O)C(C)C)ccc1O[C@@H]1CC[C@@H](NC(=O)[C@@]2(F)CNC3(CCC3)C2)C1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 748437   

TargetHistone acetyltransferase KAT2A(Human)
Pfizer

US Patent
LigandPNGBDBM748437(US20250188030, Compound C18)
Affinity DataKi:  0.100nMAssay Description:KAT2A/B Assay Protocol:A) Compound preparation1) Prepare 10 mM stock solutions in 100% DMSO from solid material.2) Serial dilute 10 mM, 1 mM, 0.1 or ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/7/2025
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B(Human)
Pfizer

US Patent
LigandPNGBDBM748437(US20250188030, Compound C18)
Affinity DataKi:  0.310nMAssay Description:KAT2A/B Assay Protocol:A) Compound preparation1) Prepare 10 mM stock solutions in 100% DMSO from solid material.2) Serial dilute 10 mM, 1 mM, 0.1 or ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/7/2025
Entry Details
US Patent