BDBM757243 US20250223284, Example Table 2.8

SMILES CC[C@@]1(O)CNC[C@@H](C(=O)N[C@H](C#N)Cc2ccc(-c3ccc4oc(=O)n(C)c4c3)cc2)OC1

InChI Key

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 757243   

TargetDipeptidyl peptidase 1(Mouse)
Insmed

US Patent
LigandPNGBDBM757243(US20250223284, Example Table 2.8)
Affinity DataIC50: 36.9nMAssay Description:Table 2: Test articles were applied to active mouse DPP1 enzyme (R&D Systems; Minneapolis, MN) in Assay Buffer (50 mM MES pH 5.5, 50 mM NaCl, 5 mM DT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/27/2025
Entry Details
US Patent