BDBM760842 1-Methyl-5-((R)-3-methyl-morpholin-4-yl)-7-(2-methyl-pyridin-3-yl)-3-(1H-pyrazol-3-yl)-1H-pyrazolo[4,3-b]pyridine ::US12371430, Compound 4
SMILES Cc1ncccc1-c1cc(N2CCOC[C@H]2C)nc2c(-c3cc[nH]n3)nn(C)c12
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 760842
Affinity DataIC50: 0.800nMAssay Description:The ATR/ATRIP enzymatic assay is performed as a TR-FRET-(HTRF™, Cisbio Bioassays) based 384-well assay. In a first step, purified human recombinant A...More data for this Ligand-Target Pair
