BDBM763796 2-(8-methoxy-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-3,4-dimethyl-6-(1-(tetrahydro-2H-pyran-4-yl)piperidin-3-yl)-9H-carbazole::US12384760, Example 28

SMILES COc1cc(-c2cc3[nH]c4ccc(C5CCCN(C6CCOCC6)C5)cc4c3c(C)c2C)cn2ncnc12

InChI Key InChIKey=XSDKQSKIEHNLAS-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 763796   

TargetToll-like receptor 8(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 763796BDBM763796(2-(8-methoxy-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-3...)
Affinity DataIC50: 0.700nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetToll-like receptor 7(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 763796BDBM763796(2-(8-methoxy-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-3...)
Affinity DataIC50: 7.80nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetToll-like receptor 9(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 763796BDBM763796(2-(8-methoxy-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-3...)
Affinity DataIC50: 523nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent