BDBM763798 2-(8-methoxy-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-3,4-dimethyl-6-(1-(2-(methylsulfonyl)ethyl)azetidin-3-yl)-9H-carbazole::US12384760, Example 30

SMILES COc1cc(-c2cc3[nH]c4ccc(C5CN(CCS(C)(=O)=O)C5)cc4c3c(C)c2C)cn2ncnc12

InChI Key InChIKey=YVZPHYGTFNBMCP-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 763798   

TargetToll-like receptor 8(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 763798BDBM763798(2-(8-methoxy-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-3...)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetToll-like receptor 7(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 763798BDBM763798(2-(8-methoxy-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-3...)
Affinity DataIC50: 5.5nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetToll-like receptor 9(Human)
Bristol-Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 763798BDBM763798(2-(8-methoxy-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-3...)
Affinity DataIC50: 813nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent