BDBM764014 US12384776, Compound D133

SMILES CNC(=O)N1CCc2c(-c3cc(OC)c(CN4CC5(CC(C#Cc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)c(OC)c3)cn(C)c(=O)c2C1

InChI Key InChIKey=KBXNYSXZKYQXIH-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 764014   

TargetBromodomain-containing protein 9(Human)
Foghorn Therapeutics

US Patent
LigandPNGBDBM764014(US12384776, Compound D133)
Affinity DataIC50: 10nMAssay Description:A stable SYO-1 cell line expressing 3×FLAG-NLuc-BRD9 was generated. On day 0 cells were seeded in 30 μL media into each well of 384-well cell culture...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
Go to US Patent