BDBM771613 US20250084112, Example 4A

SMILES Cc1cc(OC(F)(F)F)ccc1N1CN(c2ccc(=O)[nH]c2C)C(=O)c2cc(C(F)(F)F)cnc21

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 771613   

TargetSodium channel protein type 10 subunit alpha(Human)
Glaxosmithkline Intellectual Property Development

US Patent
LigandPNGBDBM771613(US20250084112, Example 4A)
Affinity DataIC50: 31.6nMAssay Description:Human embryonic kidney 293 cells (HEK293) expressing human Nav1.8, human Navβ1 and human TREK1 (HEK293-Nav1.8) were grown at 37° C., 5% CO2 in 150 cm...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
12/30/2025
Entry Details
US Patent