BDBM773958 US20250302837, Example TY-51469

SMILES Cc1c(S(=O)(=O)Nc2ccc(-c3nc(C(=O)O)cs3)cc2S(C)(=O)=O)sc2ccc(F)cc12

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 773958   

TargetChymase(Human)
Socpra Sciences Sante Et Humaines S.E.C.

US Patent
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 20nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

Targetchymase(Golden hamster)
Socpra Sciences Sante Et Humaines S.E.C.

US Patent
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 66nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetCathepsin G(Human)
Socpra Sciences Sante Et Humaines S.E.C.

US Patent
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 1.30E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetPlasma kallikrein(Human)
Socpra Sciences Sante Et Humaines S.E.C.

US Patent
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 2.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetPlasminogen(Human)
Socpra Sciences Sante Et Humaines S.E.C.

US Patent
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 2.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetCoagulation factor X(Human)
Socpra Sciences Sante Et Humaines S.E.C.

US Patent
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 2.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetTissue-type plasminogen activator(Human)
Socpra Sciences Sante Et Humaines S.E.C.

US Patent
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 2.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetSerine protease 1(Human)
Socpra Sciences Sante Et Humaines S.E.C.

US Patent
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 2.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetProthrombin(Human)
Socpra Sciences Sante Et Humaines S.E.C.

US Patent
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 2.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetCoagulation factor XI(Human)
Socpra Sciences Sante Et Humaines S.E.C.

US Patent
LigandPNGBDBM773958(US20250302837, Example TY-51469)
Affinity DataIC50: 2.00E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent