BDBM773972 4-((1H- pyrazol-1- yl)methyl)-N- ((5-(tert- butyl)-2- methoxyphenyl) sulfonyl)-3- (methoxymethyl) benzamide::US20250304535, Example C12

SMILES COCc1cc(C(=O)NS(=O)(=O)c2cc(C(C)(C)C)ccc2OC)ccc1Cn1cccn1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 773972   

TargetHistone acetyltransferase KAT6B [657-1069](Human)
Beigene Switzerland

US Patent
LigandPNGBDBM773972(4-((1H- pyrazol-1- yl)methyl)-N- ((5-(tert- butyl)...)
Affinity DataIC50: 75nMAssay Description:Testing for the inhibition activities of various compounds disclosed herein was carried out at room temperature in assay buffer containing 100 mM Tri...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetHistone acetyltransferase KAT6A [497-780](Human)
Beigene Switzerland

US Patent
LigandPNGBDBM773972(4-((1H- pyrazol-1- yl)methyl)-N- ((5-(tert- butyl)...)
Affinity DataIC50: 75nMAssay Description:Testing for the inhibition activities of various compounds disclosed herein was carried out at room temperature in assay buffer containing 100 mM Tri...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent