BDBM774000 4-((4-amino-1H-pyrazol-1- yl)methyl)-N-((6-(tert- butyl)-3-methoxypyridin-2- yl)sulfonyl)-3- methoxybenzamide::US20250304535, Example C38

SMILES COc1cc(C(=O)NS(=O)(=O)c2nc(C(C)(C)C)ccc2OC)ccc1Cn1cc(N)cn1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 774000   

TargetHistone acetyltransferase KAT6B [657-1069](Human)
Beigene Switzerland

US Patent
LigandPNGBDBM774000(4-((4-amino-1H-pyrazol-1- yl)methyl)-N-((6-(tert- ...)
Affinity DataIC50: 100nMAssay Description:Testing for the inhibition activities of various compounds disclosed herein was carried out at room temperature in assay buffer containing 100 mM Tri...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetHistone acetyltransferase KAT6A [497-780](Human)
Beigene Switzerland

US Patent
LigandPNGBDBM774000(4-((4-amino-1H-pyrazol-1- yl)methyl)-N-((6-(tert- ...)
Affinity DataIC50: 100nMAssay Description:Testing for the inhibition activities of various compounds disclosed herein was carried out at room temperature in assay buffer containing 100 mM Tri...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent