BDBM774130 5-((1H-pyrazol-1- yl)methyl)-N- ((5-(8-oxa-3- azabicyclo[3.2.1] octan-3- yl)-2- methoxyphenyl) sulfonyl)- 6-methoxy- picolinamide::US20250304535, Example C62

SMILES COc1ccc(N2CC3CCC(C2)O3)cc1S(=O)(=O)NC(=O)c1ccc(Cn2cccn2)c(OC)n1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 774130   

TargetHistone acetyltransferase KAT6B [657-1069](Human)
Beigene Switzerland

US Patent
LigandChemical structure of BindingDB Monomer ID 774130BDBM774130(5-((1H-pyrazol-1- yl)methyl)-N- ((5-(8-oxa-3- azab...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetHistone acetyltransferase KAT6A [497-780](Human)
Beigene Switzerland

US Patent
LigandChemical structure of BindingDB Monomer ID 774130BDBM774130(5-((1H-pyrazol-1- yl)methyl)-N- ((5-(8-oxa-3- azab...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent