BDBM775459 US12435087, Compound I-287

SMILES C=C(C(=O)NCc1cccc([C@@H]2c3cnn(-c4ccccc4)c3N(CC)C(=O)[C@H]2NC(=O)c2ccn(C(F)(F)F)n2)c1)C(C)N1CC2CC(C1)O2

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 775459   

TargetDCN1-like protein 1(Human)
Cellarity

US Patent
LigandPNGBDBM775459(US12435087, Compound I-287)
Affinity DataIC50: 200nMAssay Description:The DCN1 protein was biotinylated (EZ sulfo-NHS-LC-biotin; Thermofisher) for labeling with streptavidin terbium (Tb) cryptate in the reaction. The pr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetDCN1-like protein 1(Human)
Cellarity

US Patent
LigandPNGBDBM775459(US12435087, Compound I-287)
Affinity DataIC50: 200nMAssay Description:The DCN1 protein was biotinylated (EZ sulfo-NHS-LC-biotin; Thermofisher) for labeling with streptavidin terbium (Tb) cryptate in the reaction. The pr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent