BDBM786863 2-(7-((2S,5R)-2,5-dimethyl-4-(1-(2-methylthieno[3,2-b]pyridin-5-yl)ethyl)piperazin-1-yl)-4-methyl-5-oxo-4,5-dihydro-2H-pyrazolo[4,3-b]pyridin-2-yl)acetonitrile::US20250346597, Compound A155a

SMILES Cc1cc2nc([C@H](C)N3C[C@H](C)N(c4cc(=O)n(C)c5cn(CC#N)nc45)C[C@H]3C)ccc2s1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 786863   

TargetDiacylglycerol kinase zeta(Human)
BEONE MEDICINES I GMBH

US Patent
LigandChemical structure of BindingDB Monomer ID 786863BDBM786863(2-(7-((2S,5R)-2,5-dimethyl-4-(1-(2-methylthieno[3,...)
Affinity DataIC50: 20nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
3/4/2026
Entry Details US Patent

TargetDiacylglycerol kinase alpha(Human)
BEONE MEDICINES I GMBH

US Patent
LigandChemical structure of BindingDB Monomer ID 786863BDBM786863(2-(7-((2S,5R)-2,5-dimethyl-4-(1-(2-methylthieno[3,...)
Affinity DataIC50: 1.14E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
3/4/2026
Entry Details US Patent