BDBM787587 3-(1-{[(1S)-2,2-Difluorocyclopropyl]methyl}-1H-pyrazol-4-yl)-8-methoxy-2-(trifluoromethyl)-4H-pyrido[1,2-a]pyrimidin-4-one::US12473289, Example 70

SMILES COc1ccn2c(=O)c(-c3cnn(C[C@@H]4CC4(F)F)c3)c(C(F)(F)F)nc2c1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 787587   

TargetAcyl-CoA (8-3)-desaturase(Human)
AMGEN INC.

US Patent
LigandChemical structure of BindingDB Monomer ID 787587BDBM787587(3-(1-{[(1S)-2,2-Difluorocyclopropyl]methyl}-1H-pyr...)
Affinity DataIC50: 10.5nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
3/8/2026
Entry Details US Patent