BDBM787659 N-ethyl-5-fluoro-N-isopropyl-2-((5-(2-(6-((2-methoxy-2-methylpropyl)amino)-2-methylhexan-3-yl)-2,6-diazaspiro[3.4]octan-6-yl)-1,2,4-triazin-6-yl)oxy)benzamide::US12473295, Compound 69

SMILES CCN(C(=O)c1cc(F)ccc1Oc1nncnc1N1CCC2(C1)CN(C(CCCNCC(C)(C)OC)C(C)C)C2)C(C)C

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 787659   

TargetHistone-lysine N-methyltransferase 2A(Human)
Janssen Pharmaceutica NV

US Patent
LigandChemical structure of BindingDB Monomer ID 787659BDBM787659(N-ethyl-5-fluoro-N-isopropyl-2-((5-(2-(6-((2-metho...)
Affinity DataIC50: 16nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
3/8/2026
Entry Details US Patent

TargetMenin(Human)
Janssen Pharmaceutica NV

US Patent
LigandChemical structure of BindingDB Monomer ID 787659BDBM787659(N-ethyl-5-fluoro-N-isopropyl-2-((5-(2-(6-((2-metho...)
Affinity DataIC50: 99nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
3/8/2026
Entry Details US Patent