BDBM788158 US12473303, Compound H-APPAMP-015

SMILES Cc1ccn2c(CNc3cc(NC[C@H]4CCNC[C@@H]4O)nc4c(C(C)C)cnn34)c(C)nc2c1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 788158   

LigandChemical structure of BindingDB Monomer ID 788158BDBM788158(US12473303, Compound H-APPAMP-015)
Ligand Info
In Depth
Date in BDB:
3/8/2026
Entry Details US Patent

TargetCyclin-K/Cyclin-dependent kinase 12(Human)
Carrick Therapeutics Limited

US Patent
LigandChemical structure of BindingDB Monomer ID 788158BDBM788158(US12473303, Compound H-APPAMP-015)
Affinity DataIC50: 277nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
3/8/2026
Entry Details US Patent