BDBM788164 US12473303, Compound H-APPAMP-021

SMILES CC(C)c1cnn2c(NCc3cnc4ccccc4c3)cc(NC[C@H]3CCNC[C@@H]3O)nc12

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 788164   

LigandChemical structure of BindingDB Monomer ID 788164BDBM788164(US12473303, Compound H-APPAMP-021)
Affinity DataIC50: 28nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
3/8/2026
Entry Details US Patent

TargetCyclin-K/Cyclin-dependent kinase 12(Human)
Carrick Therapeutics Limited

US Patent
LigandChemical structure of BindingDB Monomer ID 788164BDBM788164(US12473303, Compound H-APPAMP-021)
Affinity DataIC50: 167nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
3/8/2026
Entry Details US Patent