BDBM792349 3-(5-((3-(2-fluoro-3-(pyridin-4-yl)phenyl)-1,2,4-oxadiazol-5-yl)methyl)-2-oxobenzo[d]oxazol-3(2H)-yl)piperidine-2,6-dione::US20260042752, Compound 143::US12565492, Compound 21

SMILES O=C1CCC(n2c(=O)oc3ccc(Cc4nc(-c5cccc(-c6ccncc6)c5F)no4)cc32)C(=O)N1

InChI Key InChIKey=SAJVTDFLFRYVNN-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 792349   

LigandChemical structure of BindingDB Monomer ID 792349BDBM792349(3-(5-((3-(2-fluoro-3-(pyridin-4-yl)phenyl)-1,2,4-o...)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/13/2026
Entry Details US Patent

LigandChemical structure of BindingDB Monomer ID 792349BDBM792349(3-(5-((3-(2-fluoro-3-(pyridin-4-yl)phenyl)-1,2,4-o...)
Affinity DataEC50:  55nMAssay Description:This cell based assay measures the ability of compounds to inhibit the constitutive cAMP activity of GPR6 receptor expressed in CHO-K1 cells. CHO cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details US Patent