BDBM792352 US20260042752, Compound 146::US12565492, Compound 146

SMILES O=C1CC[C@H](n2c(=O)oc3ccc(Cc4nc(-c5ccccc5)no4)cc32)C(=O)N1

InChI Key InChIKey=XGNIJIQFXVUHJG-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 792352   

LigandChemical structure of BindingDB Monomer ID 792352BDBM792352(US20260042752, Compound 146 | US12565492, Compound...)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/13/2026
Entry Details US Patent

LigandChemical structure of BindingDB Monomer ID 792352BDBM792352(US20260042752, Compound 146 | US12565492, Compound...)
Affinity DataEC50: <10nMAssay Description:This cell based assay measures the ability of compounds to inhibit the constitutive cAMP activity of GPR6 receptor expressed in CHO-K1 cells. CHO cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details US Patent