BDBM792463 4-(4-{5-[5-fluoro-6-(2-methoxyethoxy)-1H-indazol-3-yl]-1,2-oxazol-3-yl}phenyl)-1lambda4-thiomorpholin-1-one::US20260042753, Compound A127

SMILES COCCOc1cc2[nH]nc(-c3cc(-c4ccc(N5CCS(=O)CC5)cc4)no3)c2cc1F

InChI Key InChIKey=YRFIWFZSXPHFTF-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 792463   

TargetMast/stem cell growth factor receptor Kit [V654A](Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 792463BDBM792463(4-(4-{5-[5-fluoro-6-(2-methoxyethoxy)-1H-indazol-3...)
Affinity DataIC50: 0.370nMAssay Description:This cell based assay measures the ability of compounds to inhibit the constitutive cAMP activity of GPR6 receptor expressed in CHO-K1 cells. CHO cel...More data for this Ligand-Target Pair
Target InfoPDB
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Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details US Patent