BDBM792534 5-fluoro-6-(2-methoxyethoxy)-3-(3-{4-[(1R,4R)-2-oxa-5-azabicyclo[2.2.1]heptane-5-carbonyl]phenyl}-1,2-oxazol-5-yl)-1H-indazole::US20260042753, Compound A163

SMILES COCCOc1cc2[nH]nc(-c3cc(-c4ccc(C(=O)N5C[C@H]6C[C@@H]5CO6)cc4)no3)c2cc1F

InChI Key InChIKey=APZIHRQKIVKDKP-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 792534   

TargetMast/stem cell growth factor receptor Kit [V654A](Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 792534BDBM792534(5-fluoro-6-(2-methoxyethoxy)-3-(3-{4-[(1R,4R)-2-ox...)
Affinity DataIC50: 0.540nMAssay Description:The in vitro affinity of the compounds of the present invention for the CXCR1 and CXCR2 receptors was determined on a functional test of the β-a...More data for this Ligand-Target Pair
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Ligand Info
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Date in BDB:
6/24/2026
Entry Details US Patent