BDBM792590 1-(4-{5-[5-fluoro-6-(2-methoxyethoxy)-1H-indazol-3-yl]-1,2-oxazol-3-yl}benzoyl)-3-(pyridin-3-yl)azetidin-3-ol::US20260042753, Compound A221

SMILES COCCOc1cc2[nH]nc(-c3cc(-c4ccc(C(=O)N5CC(O)(c6cccnc6)C5)cc4)no3)c2cc1F

InChI Key InChIKey=QQFCFSCOFGIWDG-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 792590   

TargetMast/stem cell growth factor receptor Kit [V654A](Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 792590BDBM792590(1-(4-{5-[5-fluoro-6-(2-methoxyethoxy)-1H-indazol-3...)
Affinity DataIC50: 0.540nMAssay Description:CaMKII activity in neonatal rat ventricular myocytes (NRVM) was measured by monitoring the phosphorylation level of phospholamban using high-content ...More data for this Ligand-Target Pair
Target InfoPDB
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Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details US Patent