BDBM794753 3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-benzo[h]quinoline-6-carbonitrile::US20260062412, Compound B26

SMILES N#Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccccc12

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 794753   

TargetMyelin transcription factor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 794753BDBM794753(3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-benz...)
Affinity DataIC50: 0.370nMAssay Description:Measurement of [Ca2+]i using a FLIPR: CHO-OX1 or CHO-OX2 cells are seeded into black-walled clear-base 384-well plates (Costar) at a density of 20,00...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/15/2026
Entry Details US Patent

TargetMyelin transcription factor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 794753BDBM794753(3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-benz...)
Affinity DataIC50: 10nMAssay Description:NIH Molecular Libraries Screening Centers Network [MLSCN] Emory Chemical Biology Discovery Center in MLSCN Assay provider: Dr. Randal Kaufman, Univer...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/15/2026
Entry Details US Patent