BDBM794865 3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1-methylpyrazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C88

SMILES Cn1cc(-c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)cn1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 794865   

TargetMyelin transcription factor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 794865BDBM794865(3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1-methylpy...)
Affinity DataIC50: 0.170nMAssay Description:Measurement of [Ca2+]i using a FLIPR: CHO-OX1 or CHO-OX2 cells are seeded into black-walled clear-base 384-well plates (Costar) at a density of 20,00...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/15/2026
Entry Details US Patent

TargetMyelin transcription factor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 794865BDBM794865(3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1-methylpy...)
Affinity DataIC50: 4.40nMAssay Description:NIH Molecular Libraries Screening Centers Network [MLSCN] Emory Chemical Biology Discovery Center in MLSCN Assay provider: Dr. Randal Kaufman, Univer...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/15/2026
Entry Details US Patent