BDBM798329 (R)-N-(2-(1-methylpyrrolidin-2-yl)-1H-pyrrolo[3,2-c]pyridin-6-yl)-5-(1H-pyrazol-4-yl)picolinamide::US20260078121, Example 2

SMILES CN1CCC[C@@H]1c1cc2cnc(NC(=O)c3ccc(-c4cn[nH]c4)cn3)cc2[nH]1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 798329   

TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Bridge Medicines

US Patent
LigandChemical structure of BindingDB Monomer ID 798329BDBM798329((R)-N-(2-(1-methylpyrrolidin-2-yl)-1H-pyrrolo[3,2-...)
Affinity DataIC50: 7nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent

TargetProtein ENL(Human)
Bridge Medicines

US Patent
LigandChemical structure of BindingDB Monomer ID 798329BDBM798329((R)-N-(2-(1-methylpyrrolidin-2-yl)-1H-pyrrolo[3,2-...)
Affinity DataIC50: 195nMAssay Description:CHO-K1 cells expressing Ga16 and hGPR120 were dispensed into each well of a 96-well plate (3×104 cells/100 μl/well) and then incubated in 5% CO2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent