BDBM798451 3-Amino-4-(7-fluoro-1H-indazol-4-yl)-8-methyl-7-(oxetan-3-yl)-1H-1,5-naphthyridin-2-one::US20260078122, Example 122

SMILES Cc1c(C2COC2)cnc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c12

InChI Key

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 798451   

LigandChemical structure of BindingDB Monomer ID 798451BDBM798451(3-Amino-4-(7-fluoro-1H-indazol-4-yl)-8-methyl-7-(o...)
Affinity DataIC50: 10nMAssay Description:The cellular potency of Compound 1 in suppressing intracellular 2-HG levels was determined in cell lines expressing five different mutated IDH-1 prot...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/29/2026
Entry Details
US Patent