BDBM801907 US12606544, Example 44::methyl (R)-6-((5-fluoro-4-(7-(3-methoxy-2-(4- methylpiperazin-1-yl)propanamido)-1H-indol-3- yl)pyrimidin-2-yl)amino)-1H-indazole-3- carboxylate
SMILES COC[C@H](C(=O)Nc1cccc2c(-c3nc(Nc4ccc5c(C(=O)OC)n[nH]c5c4)ncc3F)c[nH]c12)N1CCN(C)CC1
InChI Key InChIKey=WBWWFBNXFPMWNG-UHFFFAOYSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 801907
Affinity DataIC50: 0.270nMAssay Description:JAK1, JAK2, JAK3 and Tyk2 were purchased from Carna Biosciences, Inc. As the substrate, LANCE Ultra ULight-JAK1 Peptide (manufactured by PerkinElmer ...More data for this Ligand-Target Pair
Affinity DataIC50: 147nMAssay Description:JAK1, JAK2, JAK3 and Tyk2 were purchased from Carna Biosciences, Inc. As the substrate, LANCE Ultra ULight-JAK1 Peptide (manufactured by PerkinElmer ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:JAK1, JAK2, JAK3 and Tyk2 were purchased from Carna Biosciences, Inc. As the substrate, LANCE Ultra ULight-JAK1 Peptide (manufactured by PerkinElmer ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:JAK1, JAK2, JAK3 and Tyk2 were purchased from Carna Biosciences, Inc. As the substrate, LANCE Ultra ULight-JAK1 Peptide (manufactured by PerkinElmer ...More data for this Ligand-Target Pair