BDBM802383 US20260109697, Compound A74::[4-(1-Methyl-1H-pyrazol-4-yl)-benzyl]-{6-[7-(3-morpholin-4-yl-propoxy)-imidazo[1,2-a]pyridin-3-yl]-pyrimidin-4-yl}-amine

SMILES Cn1cc(-c2ccc(CNc3cc(-c4cnc5cc(OCCCN6CCOCC6)ccn45)ncn3)cc2)cn1

InChI Key InChIKey=CSSUJUPJGRGFRM-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 802383   

TargetMast/stem cell growth factor receptor Kit [V654A](Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 802383BDBM802383([4-(1-Methyl-1H-pyrazol-4-yl)-benzyl]-{6-[7-(3-mor...)
Affinity DataIC50: 4.80nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
Target InfoPDB
GoogleScholar
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2026
Entry Details
US Patent