BDBM802461 (4-Fluoro-6-pyrrolidin-1-yl-pyridin-3-ylmethyl)-(6-imidazo[1,2-a]pyridin-3-yl-pyrimidin-4-yl)-amine::US20260109697, Compound A152

SMILES Fc1cc(N2CCCC2)ncc1CNc1cc(-c2cnc3ccccn23)ncn1

InChI Key InChIKey=YOJOXXFZZHCQDT-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 802461   

TargetMast/stem cell growth factor receptor Kit [V654A](Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 802461BDBM802461((4-Fluoro-6-pyrrolidin-1-yl-pyridin-3-ylmethyl)-(6...)
Affinity DataIC50: 3.80nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
Target InfoPDB
GoogleScholar
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2026
Entry Details
US Patent