BDBM802573 N-{[4-(2-methyl-1,3-oxazol-4-yl)phenyl]methyl}-6-[7-(2-{4H,5H,6H,7H-[1,2,3]triazolo[1,5-a]pyrazin-5-yl}ethoxy)imidazo[1,2-a]pyridin-3-yl]pyrimidin-4-amine::US20260109697, Compound A264

SMILES Cc1nc(-c2ccc(CNc3cc(-c4cnc5cc(OCCN6CCn7nncc7C6)ccn45)ncn3)cc2)co1

InChI Key InChIKey=DPWUGBXABZFQRZ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 802573   

TargetMast/stem cell growth factor receptor Kit [V654A](Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 802573BDBM802573(N-{[4-(2-methyl-1,3-oxazol-4-yl)phenyl]methyl}-6-[...)
Affinity DataIC50: 1.60nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
Target InfoPDB
GoogleScholar
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2026
Entry Details
US Patent