BDBM805312 (S)-4-amino-7-fluoro-N- methyl-N-(6-(trifluoro- methyl)-2,3-dihydro- benzofuran-3-yl)imidazo [1,5-a]quinoxaline-8- carboxamide::US20260125380, Example 29

SMILES CN(C(=O)c1cc3c(cc1F)nc(N)c2cncn23)[C@@H]5COc4cc(C(F)(F)F)ccc45

InChI Key InChIKey=MPJUJZTYGCAZPL-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 805312   

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Shanghai Apeiron Therapeutics Company

US Patent
LigandChemical structure of BindingDB Monomer ID 805312BDBM805312((S)-4-amino-7-fluoro-N- methyl-N-(6-(trifluoro- me...)
Affinity DataIC50: 1.14E+4nMAssay Description:A panel of four LanthaScreen JAK biochemical assays (JAK1, 2, 3 and Tyk2) were carried in a common kinase reaction buffer (50 mM HEPES, pH 7.5, 0.01%...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/17/2026
Entry Details
US Patent