BDBM9040 1H-Indazole-3-carboxylic Acid [7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]amide::Indazole-Tacrine Heterodimer 23::N-{7-[(6-chloro-1,2,3,4-tetrahydroacridin-9-yl)amino]heptyl}-1H-indazole-3-carboxamide

SMILES Clc1ccc2c(NCCCCCCCNC(=O)c3n[nH]c4ccccc34)c3CCCCc3nc2c1

InChI Key InChIKey=XYRVXZVCEIJZMQ-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 9040   

TargetAcetylcholinesterase(Bovine)
Neuropharma

LigandPNGBDBM9040(1H-Indazole-3-carboxylic Acid [7-(6-Chloro-1,2,3,4...)
Affinity DataIC50:  95nMpH: 8.0 T: 30°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The absorbance changes at 405 nm were recorded for 5 min with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAcetylcholinesterase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM9040(1H-Indazole-3-carboxylic Acid [7-(6-Chloro-1,2,3,4...)
Affinity DataIC50:  95nMAssay Description:Inhibition of AChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCholinesterase(Human)
Neuropharma

LigandPNGBDBM9040(1H-Indazole-3-carboxylic Acid [7-(6-Chloro-1,2,3,4...)
Affinity DataIC50:  79nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The absorbance changes at 405 nm were recorded for 5 min with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed