BDBM50636456 Sonrotoclax::Bgb 11417::Bgb-11417::BGB-11417::BGB11417
SMILES CC(C)c1ccccc1[C@@H]1CCCN1C1CC2(CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NC[C@H]5CC[C@](C)(O)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)C1
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50636456
Affinity DataIC50: 0.0190nMAssay Description:Inhibition of Bcl-2 (unknown origin) using (Ac-GQVGRQLAIIGDK (FITC) INR-amide) as substrate preincubated for 30 mins followed by substrate addition a...More data for this Ligand-Target Pair
Affinity DataKd: 0.240nMAssay Description:Binding affinity to His-tagged Bcl-2 G101V mutant (unknown origin) by SPR methodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.340nMAssay Description:Inhibition of Bcl-2 G101V mutant (unknown origin) using (Ac-GQVGRQLAIIGDK (FITC) INR-amide) as substrate preincubated for 30 mins followed by substra...More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of Bcl-Xl (unknown origin)More data for this Ligand-Target Pair
