BDBM50212626 LY-255283

SMILES CCc1cc(C(C)=O)c(O)cc1OCCCCCC(C)(C)c1nn[nH]n1

InChI Key InChIKey=WCGXJPFHTHQNJL-UHFFFAOYSA-N

Data  1 KI  2 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50212626   

TargetLeukotriene B4 receptor 1/2(Human)TBA

LigandBDBM50212626(LY-255283)Copy SMILESCopy InChI

Affinity DataKi:  77nMAssay Description:Inhibition of specific binding of [3H]-LTB4 to LTB4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

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In Depth
Date in BDB:
9/19/2018
Entry Details
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TargetLeukotriene B4 receptor 1/2(Human)TBA

LigandBDBM50212626(LY-255283)Copy SMILESCopy InChI

Affinity DataIC50: 85nMAssay Description:Inhibition of specific binding of [3H]LTB4 to LTB4 receptor in human neutrophilsMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchasePC cidPC sidSimilars

In Depth
Date in BDB:
9/19/2018
Entry Details
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TargetLeukotriene B4 receptor 2(Human)
Incerebro

Curated by ChEMBL

LigandBDBM50212626(LY-255283)Copy SMILESCopy InChI

Affinity DataIC50: 150nMAssay Description:Displacement of [3H]LTB4 from HA-epitope tagged human BLT2 expressed in CHOK1 cells incubated for 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair

Target InfoUniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchasePC cidPC sidSimilars

In Depth
Date in BDB:
8/13/2021
Entry Details Article
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