BDBM50092155 (4S,5R)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carboxylic acid (4-bromo-phenyl)-amide::3-Oxo-4,5-diphenyl-pyrazolidine-1-carboxylic acid (4-bromo-phenyl)-amide(LY288513)::CHEMBL333081::LY-288513

SMILES Brc1ccc(NC(=O)N2NC(=O)[C@H]([C@@H]2c2ccccc2)c2ccccc2)cc1

InChI Key InChIKey=LMUQHXHWJWQXSD-PMACEKPBSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50092155   Sort by

LigandPNGBDBM50092155((4S,5R)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carboxyl...)
Affinity DataIC50:  19nMpH: 7.4Assay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type B receptor in mouse brain at a pH of 6.5More data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50092155((4S,5R)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carboxyl...)
Affinity DataIC50:  2.05E+4nMAssay Description:The compound was tested for its activity to inhibit the binding of [3H]-L-364,718 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50092155((4S,5R)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carboxyl...)
Affinity DataIC50:  31nMpH: 6.5Assay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type B receptor in mouse brain at a pH of 7.4More data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50092155((4S,5R)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carboxyl...)
Affinity DataIC50:  2.05E+4nMAssay Description:Half maximal inhibition of specific binding of [125I]-Bolton-Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50092155((4S,5R)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carboxyl...)
Affinity DataIC50:  1.16E+4nMAssay Description:The compound was tested for its activity to inhibit the binding of [3H]-L-364,718 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50092155((4S,5R)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carboxyl...)
Affinity DataIC50:  19nMAssay Description:Half maximal inhibition of specific binding of [125I]Bolton-Hunter CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed