BDBM86260 CAS_465-65-6::NALOXONE::NSC_10064::Naloxone(-)

SMILES C=CCN1CCC23c4c5ccc(O)c4OC2C(=O)CCC3(O)C1C5

InChI Key InChIKey=UZHSEJADLWPNLE-UHFFFAOYSA-N

Data  8 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 86260   

TargetMu-type opioid receptor(Rat)
University of Innsbruck

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 86260BDBM86260(Naloxone(-) | NSC_10064 | CAS_465-65-6 | NALOXONE)
Affinity DataKi:  1.63nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Adolor

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 86260BDBM86260(Naloxone(-) | NSC_10064 | CAS_465-65-6 | NALOXONE)
Affinity DataKi:  3.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Adolor

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 86260BDBM86260(Naloxone(-) | NSC_10064 | CAS_465-65-6 | NALOXONE)
Affinity DataKi:  9.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Adolor

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 86260BDBM86260(Naloxone(-) | NSC_10064 | CAS_465-65-6 | NALOXONE)
Affinity DataKi:  33nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Adolor

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 86260BDBM86260(Naloxone(-) | NSC_10064 | CAS_465-65-6 | NALOXONE)
Affinity DataKi:  66.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Adolor

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 86260BDBM86260(Naloxone(-) | NSC_10064 | CAS_465-65-6 | NALOXONE)
Affinity DataKi:  488nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2012
Entry Details Article
PubMed
TargetNociceptin receptor(Mouse)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 86260BDBM86260(Naloxone(-) | NSC_10064 | CAS_465-65-6 | NALOXONE)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2013
Entry Details
PubMed
TargetNociceptin receptor(Mouse)
Mcgill University

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 86260BDBM86260(Naloxone(-) | NSC_10064 | CAS_465-65-6 | NALOXONE)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2013
Entry Details
PubMed