BDBM60419 BDBM50295658::NAM
SMILES CCCCC\C=C/C\C=C/C\C=C/C\C=C/CCCCN1C(=O)C=CC1=O
InChI Key InChIKey=GZNZRHSGGQUYAP-DOFZRALJSA-N
Data 10 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 10 hits for monomerid = 60419
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of human recombinant MGL by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of human MGLMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Louvain Drug Research Institute
Curated by ChEMBL
Louvain Drug Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of human cerebellar membranes MAGL-like activity preincubated for 30 mins followed by 2-AG substrate addition after 90 mins by HPLC analys...More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human MAGL expressed in Escherichia coli using 6-methoxy-4-methylcoumarin ester as substrate after 3 hrs by mass spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of MAGL in rat cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of MAGL from Wistar rat brain membranes using 2-AG as substrate after 90 mins by HPLC analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of rat cerebellar membranes MAGL-like activity preincubated for 30 mins followed by 2-AG substrate addition after 90 mins by HPLC analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of FAAH in Sprague-Dawley rat brain microsomes assessed as N-(2-hydroxyethyl)-4-pyren-1-ylbutanamide conversion to 4-pyren-1-ylbutanoic ac...More data for this Ligand-Target Pair